Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,566
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2,566
R&D Systems™ AZ 13824374
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective ATAD2 bromodomain inhibitor
2,567
R&D Systems™ (-)-U-50488 hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 114528-79-9 Molecular Formula: C19H29Cl3N2O2
| CAS | 114528-79-9 |
|---|---|
| Molecular Formula | C19H29Cl3N2O2 |
2,568
R&D Systems™ CRID3 sodium salt
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent NLRP3 inflammasome inhibitor; inhibits IL-1β production
| Product Type | CRID3 sodium salt |
|---|---|
| Molecular Weight (g/mol) | 426.46 |
| Purity | 98% |
2,569
R&D Systems™ 666-15
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective CREB inhibitor
| Target | Additional Transcription Factor Compounds |
|---|---|
| CAS | 1433286-70-4 |
| Purity | >98% |
| Chemical Name or Material | 3-(3-Aminopropoxy)-N-[2-[[3-[[(4-chloro-2-hydroxyphenyl)amino]carbonyl]-2-naphthalenyl]oxy]ethyl]-2-naphthalenecarboxamide hydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C33H30ClN3O5.HCl |
| Formula Weight | 620.52 |
2,570
R&D Systems™ CLP 290
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. K+/Cl- cotransporter 2 (KCC2) activator; orally bioavailable prodrug of CLP 257 (Cat. No.5242)
| Target | KCC2 Activators |
|---|---|
| CAS | 1181083-81-7 |
| Purity | 98% |
| Chemical Name or Material | (Z)-5-Fluoro-2-((4-oxo-2-(tetrahydropyridazin-1(2 H)-yl)thiazol-5(4 H)-ylidene)methyl)phenyl pyrrolidine-1-carboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H21FN4O3S |
2,571
R&D Systems™ Ispinesib
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. High affinity and selective allosteric KSP inhibitor
| Product Type | Ispinesib |
|---|---|
| Molecular Weight (g/mol) | 517.06 |
| Purity | >98% |
2,572
R&D Systems™ MLN 4760
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective angiotensin-converting enzyme 2 (ACE2) inhibitor
2,573
R&D Systems™ Dacomitinib
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent irreversible pan ErbB inhibitor
| CAS | 1110813-31-4 |
|---|---|
| Chemical Name or Material | (2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-7-methoxy-6-quinazolinyl]-4-(1-piperidinyl)-2-butenamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C24H25ClFN5O2 |
| Formula Weight | Observed MW: 469.94 |
| Assay Percent Range | >98% |
2,574
R&D Systems™ VU 0463271
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective KCC2 inhibitor
| Target | KCC2 Inhibitors |
|---|---|
| CAS | 1391737-01-1 |
| Purity | >98% |
| Chemical Name or Material | N-Cyclopropyl-N-(4-methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C19H18N4OS2 |
| Formula Weight | 382.5 |
2,575
R&D Systems™ Hydroxy Dynasore
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Dynamin inhibitor; analog of dynasore (Cat. No. 2897)
| Product Type | Hydroxy Dynasore |
|---|---|
| Molecular Weight (g/mol) | 338.31 |
| Purity | >98% |
2,576
R&D Systems™ (R)-(-)-α-Methylhistamine dihydrobromide
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 868698-49-1 Molecular Formula: C6H13Br2N3
| CAS | 868698-49-1 |
|---|---|
| Molecular Formula | C6H13Br2N3 |
2,577
R&D Systems™ UNC 0638
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 1255517-77-1 Molecular Formula: C30H49N5O3
| CAS | 1255517-77-1 |
|---|---|
| Molecular Formula | C30H49N5O3 |
2,578
R&D Systems™ PF 3758309 dihydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent PAK4 inhibitor; orally available
| Product Type | Bioactive Small Molecule |
|---|---|
| Color | Off-white |
| Solubility | Soluble to 100mM in water and to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | PF 3758309 Dihydrochloride |
| Recommended Storage | Store at -20°C |
| Synonym | N-[(1S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide dihydrochloride |
| Molecular Formula | C25H30N8OS.2HCl |
| Formula Weight | 563.55 |
2,579
R&D Systems™ B 973B
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Positive allosteric modulator of α7 nAChRs; analgesic
| CAS | 2244989-34-0 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 3,4-Difluoro-N-[(1S)-1-[6-[4-(2-pyridinyl)-1-piperazinyl]-2-pyrazinyl]ethyl]benzenepropanamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H26F2N6O |
2,580
R&D Systems™ 1-Hex-GlcNAlk
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Metabolic chemical reporter for studying glycosylation and glycoproteins